Skip to content
BiologicalX

Comparison

CJC-1295 vs Low-Dose Naltrexone

Side-by-side of CJC-1295 and Low-Dose Naltrexone. Every row below is pulled from the compound schema and will update as our data grows. For deeper reads, follow through to each compound page.

Effects at a glance

CJC-1295

  • GHRH analog that binds the GHRH receptor on pituitary somatotrophs to release endogenous GH
  • DAC variant has ~7 day half-life via albumin binding; non-DAC variant ~30 minutes
  • Teichman 2006 trial showed sustained 2 to 10 fold IGF-1 elevation at 60 to 250 mcg/kg DAC dosing
  • Anecdotal protocols pair non-DAC CJC-1295 with Ipamorelin to mimic pulsatile GH release
  • Side effects: water retention, numbness or tingling at injection site, vivid dreams, transient flushing
  • No completed phase III RCTs; research-use-only and not FDA approved

Low-Dose Naltrexone

  • Off-label use at 1.5 to 4.5 mg, roughly one-tenth the FDA-approved 50 mg addiction-treatment dose
  • Proposed mechanisms include brief opioid receptor blockade triggering rebound endogenous opioid release, plus TLR4 antagonism
  • Compounded prescription only; insurance rarely covers; cash prices 20 to 80 USD per month
  • Younger 2013 reported ~30% pain reduction in fibromyalgia at 4.5 mg in a small crossover trial
  • Smith 2011 reported endoscopic improvement in active Crohn's disease (n=40 placebo-controlled)
  • Vivid dreams affect 20 to 40% in first 2 weeks; manageable by switching to morning dosing

Side-by-side

Attribute CJC-1295 Low-Dose Naltrexone
Category peptide pharmaceutical
Also known as CJC-1295 DAC, CJC-1295 no-DAC, Mod GRF 1-29, tesamorelin analog LDN, naltrexone (low dose)
Half-life (hr) 168 4
Typical dose (mg) 0.1 4.5
Dosing frequency weekly (DAC); 1-3x daily (non-DAC) once daily, typically at bedtime
Routes subcutaneous oral
Onset (hr) 1 1
Peak (hr) 3 1.5
Molecular weight 3367.83 341.4
Molecular formula C152H252N44O42 C20H23NO4
Mechanism Binds the GHRH receptor on pituitary somatotrophs, stimulating pulsatile growth-hormone release. The DAC modification extends plasma residence by tethering the peptide to serum albumin via a maleimide-cysteine bond. Brief mu-opioid receptor antagonism proposed to trigger compensatory upregulation of endogenous opioids; secondary TLR4 antagonism on microglia and immune cells contributes to anti-inflammatory effect.
Legal status Not FDA approved; research-use-only grey market; banned by WADA Off-label compounded prescription (naltrexone is FDA approved for opioid and alcohol use disorder at 50 mg)
WADA status banned allowed
DEA / Rx Not FDA approved; not scheduled; research-chemical status Rx only (not a controlled substance)
Pregnancy Insufficient data; not recommended Insufficient data; not routinely recommended
CAS 446262-90-4 16590-41-3
PubChem CID 91971820 5360515
Wikidata Q5012154 Q426444

Safety profile

CJC-1295

Common side effects

  • injection-site reactions
  • water retention
  • numbness or tingling at injection site
  • vivid dreams
  • transient flushing
  • head pressure or mild headache

Contraindications

  • pregnancy
  • active malignancy
  • diabetic retinopathy (theoretical)
  • history of pituitary tumor

Interactions

  • Ipamorelin: synergistic GH release; commonly co-administered in anecdotal protocols(minor)
  • insulin: GH-induced insulin resistance can shift glycemic control over weeks(moderate)
  • corticosteroids: blunt GH-axis response; reduce expected efficacy(moderate)

Low-Dose Naltrexone

Common side effects

  • vivid dreams
  • sleep disruption
  • headache
  • mild GI upset
  • fatigue (early)

Contraindications

  • concurrent opioid use
  • acute hepatitis or liver failure
  • opioid dependence
  • pregnancy (insufficient data)

Interactions

  • opioid analgesics (oxycodone, morphine, codeine): blocks analgesic effect; precipitates withdrawal in dependent users(major)
  • tramadol: blocks opioid component of analgesia(major)
  • thyroid hormone replacement: may alter dose requirements after immune modulation; monitor TSH(minor)

Which Should You Take?

Low-Dose Naltrexone comes out ahead for most readers on the criteria we weight: 2 catalogued goals, prescription-only, oral dosing, with a Tier-A outcome catalogued. CJC-1295 is the right call when one of the conditionals below applies.

Edge case: If you cannot self-administer injections, Low-Dose Naltrexone is the only oral option in this pair.

Default choice: Low-Dose Naltrexone. Wider use case, a Tier-A evidence outcome catalogued, and broader goal coverage. Reach for CJC-1295 only if your priority sits squarely in the goals it owns above.

This verdict is generated from each compound's schema (goals, legal status, evidence outcomes, dosing route). It updates automatically as our compound data evolves; the deeper read sits on each individual compound page.

Common questions

What is the difference between CJC-1295 and Low-Dose Naltrexone?

CJC-1295 and Low-Dose Naltrexone differ in category (peptide vs pharmaceutical), mechanism, and typical dosing. See the side-by-side table for full details.

Which has a longer half-life, CJC-1295 or Low-Dose Naltrexone?

CJC-1295 half-life is 168 hours; Low-Dose Naltrexone half-life is 4 hours.

Can you stack CJC-1295 with Low-Dose Naltrexone?

Stack compatibility depends on mechanism overlap, legal status, and individual response. Check each compound page for specific interactions and contraindications before combining.

Go deeper