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Comparison

Creatine Monohydrate vs Modafinil

Side-by-side of Creatine Monohydrate and Modafinil. Every row below is pulled from the compound schema and will update as our data grows. For deeper reads, follow through to each compound page.

Effects at a glance

Creatine Monohydrate

  • Increases anaerobic strength and power output by ~5 to 15% across multiple training studies
  • Adds ~1 to 2 kg of lean body mass over 4 to 12 weeks, partly intracellular water and partly true tissue gain
  • Improves 1-rep max on bench and squat by ~5 to 10% versus placebo in resistance-trained adults
  • Cognitive benefit appears mainly under sleep deprivation or high mental load, less so in well-rested individuals
  • Saturation reached in ~28 days at 3 to 5 g/day, or ~5 to 7 days with a 20 g/day loading phase
  • No evidence of renal harm in healthy adults across long-term studies; caution in pre-existing severe renal disease

Modafinil

  • FDA approved in 1998 for narcolepsy, with later additions for shift-work sleep disorder and OSA residual sleepiness
  • Schedule IV controlled substance in the US; prescription-only in EU, UK, Australia
  • Increases wakefulness via weak dopamine reuptake inhibition plus histaminergic, noradrenergic, and orexinergic activation
  • Long half-life of 12 to 15 hours requires morning dosing to avoid sleep disruption
  • Modest cognitive enhancement signal in non-sleep-deprived adults at 100 to 200 mg (Battleday meta-review 2015)
  • Substantial CYP3A4 induction reduces hormonal contraceptive efficacy; barrier methods recommended

Side-by-side

Attribute Creatine Monohydrate Modafinil
Category supplement pharmaceutical
Also known as creatine Provigil, Modalert, Modvigil, diphenylmethylsulfinyl-acetamide
Half-life (hr) 3 13
Typical dose (mg) 5000 200
Dosing frequency daily daily, morning
Routes oral oral
Onset (hr) 168 1
Peak (hr) - 3
Molecular weight 149.15 273.35
Molecular formula C4H9N3O2 C15H15NO2S
Mechanism Donates a phosphate group to ADP via creatine kinase, regenerating ATP during high-intensity, short-duration efforts. Weak dopamine reuptake inhibition plus downstream activation of histaminergic, noradrenergic, and orexinergic wake-promoting systems.
Legal status Dietary supplement (most jurisdictions) Schedule IV (US); prescription-only globally; not a supplement
WADA status allowed banned
DEA / Rx OTC supplement Schedule IV
Pregnancy Insufficient data Not recommended
CAS 57-00-1 68693-11-8
PubChem CID 586 4236
Wikidata Q408389 Q422968

Safety profile

Creatine Monohydrate

Common side effects

  • water retention
  • mild GI upset at loading doses
  • weight gain (2 to 4 lb from intracellular water)

Contraindications

  • severe renal impairment

Interactions

  • caffeine (high-dose acute): mixed data on ergogenic interference; chronic use appears compatible(minor)
  • nephrotoxic drugs (NSAIDs, cyclosporine): theoretical additive renal strain in at-risk patients(moderate)

Modafinil

Common side effects

  • headache
  • nausea
  • anxiety
  • insomnia (with late-day dosing)
  • dry mouth
  • mild blood pressure elevation

Contraindications

  • recent myocardial infarction
  • unstable angina
  • left ventricular hypertrophy
  • significant arrhythmia
  • history of Stevens-Johnson syndrome
  • psychotic disorders
  • pregnancy
  • concurrent MAOI use

Interactions

  • hormonal contraceptives: CYP3A4 induction reduces contraceptive efficacy; use barrier method(major)
  • cyclosporine: reduced cyclosporine levels via CYP3A4 induction(major)
  • warfarin: CYP2C9 inhibition raises INR(moderate)
  • phenytoin: CYP2C19 inhibition raises phenytoin levels(moderate)
  • MAOIs: potential hypertensive reaction(major)
  • classical stimulants (amphetamine, methylphenidate): additive cardiovascular and sleep-disruption effects(moderate)

Which Should You Take?

Creatine Monohydrate comes out ahead for most readers on the criteria we weight: 3 catalogued goals, OTC dietary supplement, oral dosing, with a Tier-A outcome catalogued. Modafinil is the right call when one of the conditionals below applies.

Edge case: If you want to avoid controlled substance, Creatine Monohydrate is the more accessible choice.

Default choice: Creatine Monohydrate. Lower friction to source, a Tier-A evidence outcome catalogued, and broader goal coverage. Reach for Modafinil only if your priority sits squarely in the goals it owns above.

This verdict is generated from each compound's schema (goals, legal status, evidence outcomes, dosing route). It updates automatically as our compound data evolves; the deeper read sits on each individual compound page.

Common questions

What is the difference between Creatine Monohydrate and Modafinil?

Creatine Monohydrate and Modafinil differ in category (supplement vs pharmaceutical), mechanism, and typical dosing. See the side-by-side table for full details.

Which has a longer half-life, Creatine Monohydrate or Modafinil?

Creatine Monohydrate half-life is 3 hours; Modafinil half-life is 13 hours.

Can you stack Creatine Monohydrate with Modafinil?

Stack compatibility depends on mechanism overlap, legal status, and individual response. Check each compound page for specific interactions and contraindications before combining.

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